Frontmatter -- PREFACE -- CONTENTS -- SECTION 1: STEROID HORMONE ANTAGONISTS -- STEROID AGONISTS AND ANTAGONISTS: MOLECULAR CONFORMATION, RECEPTOR BINDING AND ACTIVITY / Duax, William L. / Griffin, Jane F. / Rohrer, Douglas C. / Weeks, Charles M. -- ANTIHORMONAL ACTIVITIES OF STEROIDS WITH MODIFIED RINGS A OR B / Starka, Lubos / Hampl, Richard -- ANTAGONISM OF STEROID HORMONES BY SPECIFIC ANTIBODIES / Vecsei, Paul / Haack, Doris / Gless, Kurt-Holger -- ANTAGONISM OF STEROID HORMONE ACTION BY INTERFERENCE OF RECEPTOR FUNCTION WITH LOW MOLECULAR WEIGHT INHIBITORS / Sato, Bunzo / Nishizawa, Yasuko / Maeda, Yoshiaki / Noma, Keizo / Yamamura, Matsumoto / Yamamura, Yuichi -- ANTI-STEROIDS AND ANIMAL BEHAVIOUR : A REVIEW / Fabre-Nys, Claude -- AGONISTIC AND ANTAGONISTIC PROPERTIES OF CLOMIPHENE / Clark, James H. / Guthrie, Sylvia C. / McCormack, Shirley A. / Markavarich, Barry M. -- HYDROXYLATED ANTIOESTROGENS: NEW PHARMACOLOGICAL PROBES TO INVESTIGATE OESTROGEN AND ANTIOESTROGEN ACTION / Jordan, V. Craig -- Biological Actions and Binding Properties of a New Estrogen Antagonist / Black, Larry J. -- BINDING PROPERTIES AND LIGAND SPECIFICITY OF AN INTRACELLULAR BINDING SITE WITH SPECIFICITY FOR SYNTHETIC OESTROGEN ANTAGONISTS OF THE TRIPHENYLETHYLENE SERIES / Sutherland, Robert L. / Watta, Colin K.W. / Murphy, Leigh C. -- ESTROGEN RECEPTOR BINDING PARAMETERS OF THE HIGH AFFINITY ANTIESTROGEN 3H-H1285 / Ruh, Thomas S. / Keene, Jeffery L. / Ross, Patrick -- POTENTIAL ANTIOESTROGENIC AND ANTITUMOUR MECHANISMS OF TAMOXIFEN ACTION IN BREAST CANCER / Nicholson, Robert I. / Daniel, Paul / Syne, Joy S. / Davies, Peter -- ANTI-TUMOR ACTION OF NON-STEROIDAL ANTIESTROGENS / Sekiya, S. / Inaba, N. / Takamizawa, H. -- PROGESTERONE INHIBITION OF NUCLEAR ESTROGEN RECEPTOR RETENTION / Leavitt, Wendell W. / Evans, Rawden W. / Okulicz, William C. / McDonald, Richard G. / Hendry, William J. / Robidoux, William F. -- ADVANCES IN THE STUDY OF ANTIPROGESTATIONAL AGENTS / Kendle, K.E. -- PHARMACOLOGICAL AND CLINICAL EFFECTS OF ANT IANDROGENS / Neri, Rudolph / Kassen, Nadim -- MECHANISM OF ACTION OF A STEROIDAL ANTI-ANDROGEN TSAA-291, 16B-ETHYL-176-H YDROXYESTR-4-EN-3-ONE / Nakayama, Ryo / Hiraga, Kentaro / Miki, Takuichi -- STRUCTURE-AFFINITY RELATIONSHIP OF ANTIMINERALOCORTICOID ACTIVE STEROIDS / Wambach, Gerhard / Helber, Albert -- PROGESTIN ANTAGONISM OF ALDOSTERONE ACTION IN THE KIDNEY / Agarwal, M. K. -- CLINICAL PHARMACOLOGY AND THERAPEUTIC USE OF ALDOSTERONE ANTAGONISTS / Ramsay, Lawrence E. -- ANTIGLUCOCORTICOIDS: DIFFERENTIAL ANTAGONISM OF IN VIVO RESPONSES TO DEXAMETHASONE / Naylor, Paul H. / Rosen, Fred -- ANTAGONISM OF GLUCOCORTICOID ACTION IN VIVO / Agarwal, M. K. -- DISCRIMINATION BETWEEN GLUCOCORTICOID AGONISTS AND ANTAGONISTS BY MEANS OF RECEPTOR BINDING STUDIES / Bell, Philip A. / Jones, T. Ryland -- ANTAGONISM OF GLUCOCORTICOID ACTION BY INSULIN / Cake, Max H. / Ho, Kevin K.W. / Yeoh, George C.T. -- INHIBITION OF ADRENAL STEROID BIOSYNTHESIS BY METYRAPONE / Sonino, Nicoletta -- SECTION 2: PEPTIDE HORMONE ANTAGONISTS -- STRUCTURAL, CONFORMATIONAL AND DYNAMIC CONSIDERATIONS IN THE DEVELOPMENT OF PEPTIDE HORMONE ANTAGONISTS / Hruby, Victor J. / Mosberg, Henry I. -- INHIBITORS OF THE RENIN-ANGIOTENSIN SYSTEM / Yamamoto, Kenjiro / Miura, Katsuyuki / Abe, Youichi / Komori, Tadamitsu / Yoshimoto, Shinobu -- ANTI-PROLACTIN AND ANTI-GROWTH HORMONE RECEPTOR ANTIBODIES, AND THEIR USE AS ANTI-HORMONAL AGENTS / Waters, M.J. / Friesen, H.G. -- CLINICAL APPLICATIONS OF PROLACTIN LOWERING DRUGS / Ferrari, Carlo / Benco, Rosanna / Rampini, Pietro -- RECEPTOR ANTAGONISTS OF THE ACTIONS OF GASTROINTESTINAL PEPTIDES ON PANCREATIC ACINAR CELLS / Gardner, Jerry D. / Jensen, Robert T. -- GASTHIN ANTAGONISM / Hirst, Barry H. -- ANTIGONADAL EFFECTS OF GONADOTROPIN-RELEASING HORMONE AND AGONIST ANALOGS / Harwood, James P. / Catt, Kevin J. -- ANTAGONISTS OF HYPOTHALAMIC REGULATORY PEPTIDES AND DOPAMINE / Denef, Cali / Andries, Maria -- LUTEINIZING HORMONE RELEASING HORMONE ANALOGS AS ANTIHORMONES / Bex, Frederick / Corbin, Alan -- ANTIGONADOTROPIC, ANTISTEROIDOGENIC AND ANTISTEROIDAL ACTIVITIES OF AGONIST ANALOGS OF LUTEINIZING HORMONERELEASING HORMONE AS REVEALED BY THEIR ANTIREPRODUCTIVE ACTIVITIES / Vickery, Brian H. -- SECTION 3: MISCELLANEOUS HORMONES AND ANTAGONISTS -- HORMONAL INHIBITION OF ADENYLATE CYCLASE: A POSSIBLE MECHANISM FOR PHYSIOLOGICAL ANTAGONISM / Limbird, Lee E. -- NALOXONE AND NALTREXONE: Endorphin Antihormones / Gold, Mark S. / Pottash, A. Carter -- ANTIHISTAMINES / Dry, J. / Pradalier, A. -- X-RAY CRYSTALLOGRAPHIC STUDIES OF THYROID HORMONE, ANALOGUE AND COMPETITOR BINDING INTERACTIONS WITH HUMAN SERUM PREALBUMIN / Oatley, Stuart J. / Burridge, Jane M. / Blake, Colin C.P. -- ANTIPHEROMONES? / Baillet, Jack / Paillard, Jacques -- AUTHOR INDEX -- SUBJECT INDEX -- Backmatter
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